Therapeutics
Details checkedClinical trial listing onlyHistorical/discontinuedCheckedpublication

Neramexane by Merz

Also known as: Neramexane, Neramexane Mesylate, neramexane-mesylate, MRZ 92579, MRZ 92579-0508/1, MRZ 92579/TI/3001, NCT00405886, NCT00827008, NCT00955799, NCT00772980, NCT00739635

Merz Pharmaceuticals GmbH

Primary source
Company
Merz Pharmaceuticals GmbH
Program Type
Therapeutic
Modality
Small Molecule
Stage
Phase 3
Status
Completed
Target Gene
Route / Mode
Oral tablets
Confidence
86%
Status Confidence
Status needs checking
Evidence Strength
Needs more support
Last Reviewed
2026-06-09
Geography
Austria, Belgium, Brazil, Czechia, France, Germany, Mexico, Netherlands, Poland, Portugal, South Africa, Spain, United Kingdom, United States
Population
adult, tinnitus
Trial IDs
5
Mechanism

Oral small-molecule antagonist at NMDA receptors and alpha9/alpha10 nicotinic acetylcholine receptors evaluated for subjective tinnitus.

Indications
Notes

Merged the generated Neramexane and Neramexane Mesylate rows into one Merz-sponsored tinnitus program. The Phase 2 publication and registry identify neramexane/neramexane mesylate as the same oral tinnitus candidate; subsequent Phase 3 tinnitus studies used the mesylate name. All identified tinnitus studies are completed or terminated, and no current active Merz development signal was confirmed in this pass.

Evidence & Sources
7 structured sources
publication
Supports: canonicalName, aliases, company, modality, mechanism, indications, stage, status...
IDs: NCT00405886, neramexane mesylate
Open
registry mirror
Supports: company, stage, status, route, populationTags, geography, trialIds, keyEvents
IDs: NCT00405886, MRZ 92579-0508/1
Open
clinicaltrials
Supports: company, stage, status, route, populationTags, geography, trialIds
IDs: NCT00405886
Open
clinicaltrials
Supports: aliases, company, stage, status, route, geography, trialIds
IDs: NCT00827008
Open
clinicaltrials
Supports: aliases, company, stage, status, route, geography, trialIds
IDs: NCT00955799
Open
clinicaltrials
Supports: aliases, company, stage, status, route, geography, trialIds
IDs: NCT00772980
Open
clinicaltrials
Supports: aliases, company, stage, status, route, geography, trialIds
IDs: NCT00739635
Open
Key Events
Clinical Trials (5)
Data Checks
historical-completed-programmerged-generated-salt-name-recordsnot-confirmed-current-active-development
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